Steroids and derivatives
Medchemexpress LLC Bazedoxifene acetate | 198481-33-3 | 99.9% | C32H38N2O5 | 1 ML
Bazedoxifene acetate is an oral, nonsteroidal selective estrogen receptor modulator (SERM) primarily used as a laboratory chemical for research, especially concerning osteoporosis and pancreatic cancer. It functions as an inhibitor of IL-6/GP130 protein-protein interactions and is stable under recommended storage conditions.
- Oral, nonsteroidal selective estrogen receptor modulator (SERM)
- Inhibits ERα with IC50 of 23 nM and ERβ with IC50 of 99 nM
- Utilized for research on osteoporosis
- Functions as an inhibitor of IL-6/GP130 protein-protein interactions
- Suitable for pancreatic cancer research
- Appears as a solid
- Stable under recommended storage conditions
Medchemexpress LLC Ergocalciferol | 50-14-6 | >99.1% | 396.65 | 5 G
Vitamin D2 (Ergocalciferol) is a form of Vitamin D derived from plant sources or dietary supplements. It is used as a supplement of Vitamin D. This product is intended for research use only.
- Derived from plant sources or dietary supplements
- Activator of Vitamin D receptor
- Used as a supplement of Vitamin D
- Intended for research use
Selleck Chemical LLC Fluocinolone Acetonide 100mg 67-73-2 Flucort-N
Fluocinolone Acetonide (Flucort-N) is a corticosteroid that binds to the cytosolic glucocorticoid receptor. *For Research & Development use only. Product is not intended for drug, household, or human consumption.
Medchemexpress LLC Glepaglutide acetate | 99.5% | 4376.06 | 25 MG
Glepaglutide acetate is a long-acting GLP-2 analogue and a potent GLP-2R agonist. It reduces faecal output and increases intestinal absorption. Glepaglutide acetate alleviates small intestinal inflammation.
- Can be used in research of inflammatory bowel disease (IBD)
- Can be used in research of Crohn's disease
- Reduces faecal output
- Increases intestinal absorption
- Alleviates small intestinal inflammation
Medchemexpress LLC Bazedoxifene (acetate)-D | 198481-33-3 | C32H38N2O5 | 5 MG
Bazedoxifene (acetate)-D is the D-crystal form compound of Bazedoxifene acetate, an orally active, nonsteroidal selective estrogen receptor modulator (SERM). It targets the Estrogen Receptor/ERR pathway, specifically the Vitamin D Related/Nuclear Receptor, with IC50s of 23 nM for ERα and 99 nM for ERβ.
- D-crystal form compound
- Orally active, nonsteroidal selective estrogen receptor modulator (SERM)
- Targets estrogen receptor/ERR
- Part of vitamin D related/nuclear receptor pathway
- IC50s of 23 nM for ERα and 99 nM for ERβ
TARGETMOL CHEMICALS INC Estrone sulfate sodium 25MG
Also available in 2 mg, 5 mg, 10 mg, 50 mg and bulk. Please contact Fisher for quotes. Estrone sulfate sodium (17beta-Estrone 3-sulfate) is an endogenous steroid and an estrogen ester that is biologically inactive. It is converted by steroid sulfatase into estrone . Estrone sulfate sodium has been investigated as a ligand for targeting organic anion transporting polypeptides f Purity 98%
Apexbio Technology LLC Fluorometholone Acetate 3801-06-7 50mg
Fluorometholone Acetate (CAS 3801-06-7) is a synthetic glucocorticoid corticosteroid designed for the modulation of inflammatory responses Acting through binding to the glucocorticoid receptor it regulates the transcription of anti-inflammatory proteins while suppressing pro-inflammatory gene expression This compound is extensively utilized in ophthalmic research for modeling and investigating steroid-responsive inflammatory processes in ocular tissues Its application facilitates the study of corticosteroid-mediated pathways in eye inflammation and aids in the evaluation of anti-inflammatory interventions in preclinical settings
Medchemexpress LLC N-(1-phenylethyl)-2-(piperazin-1-yl)quinazolin-4-amine | 662164-09-2 | MFCD04077665 | 99.5% | 333.43 g/mol | C20H23N5 | 50MG
D3-βArr (N-(1-phenylethyl)-2-(piperazin-1-yl)quinazolin-4-amine; CAS 662164-09-2) is a small-molecule thyroid-stimulating-hormone (TSH) receptor modulator supplied as a high-purity solid for research use. It is provided in laboratory-scale quantities suitable for biochemical and cellular assays investigating TSH receptor pharmacology.
- High reported purity (99.5%).
- Solid form, white to off-white, suitable for standard storage.
- Molecular weight 333.43 g/mol and formula C20H23N5.
- Supplied in a 50 mg laboratory-scale quantity.
- Intended for research use only; not for human or clinical use.
- Suitable for biochemical and cellular assays targeting TSH receptor activity.
Apexbio Technology LLC Cyproterone Acetate 427-51-0 250mg
Cyproterone Acetate (CAS 427-51-0) is a small-molecule antagonist targeting the androgen receptor (AR) It is designed to inhibit AR activation thereby suppressing androgen-mediated cellular signaling Cyproterone Acetate exerts its biological activity primarily through competitive binding to AR displacing endogenous androgen ligands and blocking receptor activation and downstream signaling In experimental assays Cyproterone Acetate demonstrates AR inhibition with an IC50 value of approximately 7 1 nM At higher concentrations (EC50 around 4 0 M) it may also exhibit partial agonist activity on the AR pathway Based on these pharmacological properties Cyproterone Acetate holds research potential in studies of androgen-dependent biological processes AR signaling mechanisms and hormone-sensitive pathologies such as prostate cancer or androgen-related metabolic conditions
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eMolecules 184582-91-0 | DMPAC-Chol | Broadpharm514.839 | C33H58N2O2 | 0.000 | CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@H](CC[C@]4(C)[C@H]3CC[C@]12C)OC(=O)NCCCN(C)C | 5mg | 779524214
DMPAC-Chol | Broadpharm | 184582-91-0514.839 | C33H58N2O2 | 0.000 | CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@H](CC[C@]4(C)[C@H]3CC[C@]12C)OC(=O)NCCCN(C)C | 5mg | 779524214